Dataset: Anticancer properties of distinct antimalaria drug classes
Background: Antimalarials have anticancer potential. Results: We have systematically tested five distinct antimalaria drugs in a panel...
Background: Antimalarials have anticancer potential. Results: We have systematically tested five distinct antimalaria drugs in a panel of cancer cell lines. Conclusion: Three antimalarial classes display potent antiproliferative activity, and their potency is correlated with cancer cell gene expression patterns. Significance: We confirm and extend anticancer potential of these antimalarials and we discuss their therapeutic potential based on clinical data. Key words: Malaria, Anticancer drug, Drug Discovery, Genomics, Gene Expression, Bioinformatics, Cancer Affymetrix® HG-U133 Plus 2.0 mRNA expression arrays were used to determine the expression. CEL result files were pre-processed using the RMA (Irizarry et al, 2003) algorithm. This microarray analysis was performed for 91 cell lines.
- Species:
- human
- Samples:
- 91
- Source:
- E-GEOD-51739
- Updated:
- Dec.12, 2014
- Registered:
- Jul.11, 2014
Sample | ORIGIN | DIFFERENTIATION | AGE | CELL LINE | SEX |
---|---|---|---|---|---|
GSM1251860 | primary | not known | 72 | 1752 | male |
GSM1251859 | primary | poor | 56 | 269 | male |
GSM1251858 | not known | not known | 32 | KCL-22 | female |
GSM1251857 | not known | poor | Not available | PC-3M | male |
GSM1251856 | not known | poor | 11 | Raji | male |
GSM1251855 | not known | not known | 62 | NCI-H929 | female |
GSM1251854 | primary | not known | 51 | 486 | female |
GSM1251853 | metastasis | not known | 22 | 276 | male |
GSM1251852 | primary | not known | 55 | 698 | male |
GSM125185 | not known | not known | 59 | KG-1 | male |
GSM1251850 | primary | poor | 60 | 251 | male |
GSM1251849 | primary | moderate | 70 | 94 | male |
GSM1251848 | not known | not known | 73 | JURL-MK1 | male |
GSM1251847 | metastasis | good | 70 | 546 | male |
GSM1251846 | metastasis | poor | 63 | 289 | male |
GSM1251845 | metastasis | poor | 58 | 526 | male |
GSM1251844 | not known | poor | Not available | NCI-H460 | male |
GSM1251843 | primary | poor | 19 | MOLT-4 | male |
GSM1251842 | not known | not known | 11 | Saos-2 | female |
GSM125184 | primary | poor | 56 | 1121 | female |
GSM1251840 | recurrent | poor | 43 | 1781 | male |
GSM1251839 | metastasis | not known | 41 | 520 | male |
GSM1251838 | metastasis | not known | 35 | 1341 | female |
GSM1251837 | not known | not known | 60 | NIH:OVCAR-3 | female |
GSM1251836 | primary | not known | 74 | 1183 | male |
GSM1251835 | not known | poor | 53 | K-562 | female |
GSM1251834 | not known | poor | 69 | MCF-7 | female |
GSM1251833 | not known | not known | 81 | T-24 | female |
GSM1251832 | not known | poor | Not available | IM-9 | female |
GSM125183 | metastasis | not known | 63 | 462 | male |
GSM1251830 | not known | not known | 24 | PL-21 | male |
GSM1251829 | not known | poor | Not available | RKO | Not available |
GSM1251828 | metastasis | good | 51 | 401 | female |
GSM1251827 | not known | poor | Not available | HCT-116 | male |
GSM1251826 | not known | poor | 51 | MDA-MB-231 | female |
GSM1251825 | not known | poor | 14 | Jurkat | male |
GSM1251824 | primary | good | 76 | 899 | female |
GSM1251823 | not known | not known | 56 | lp-1 | female |
GSM1251822 | not known | poor | 36 | HL-60 | female |
GSM125182 | not known | poor | 44 | HT-29 | female |
GSM1251820 | metastasis | moderate | 60 | 1657 | female |
GSM1251819 | primary | good | 66 | 575 | male |
GSM1251818 | primary | not known | 55 | MEG-01 | male |
GSM1251817 | not known | poor | Not available | 22Rv1 | male |
GSM1251816 | not known | poor | 69 | DU-145 | male |
GSM1251815 | not known | not known | 56 | CAL-27 | male |
GSM1251814 | not known | poor | 37 | U-937 | male |
GSM1251813 | not known | not known | 7 | TE671 | female |
GSM1251812 | primary | not known | 5 | EM-2 | female |
GSM12518 | metastasis | poor | 66 | 1138 | female |
GSM1251810 | metastasis | poor | 52 | 1352 | male |
GSM1251809 | recurrent | poor | 73 | 1118 | female |
GSM1251808 | metastasis | poor | Not available | 1218 | female |
GSM1251807 | not known | not known | 31 | NOMO-1 | female |
GSM1251806 | not known | good | 53 | HUT-78 | male |
GSM1251805 | not known | not known | 56 | PANC-1 | male |
GSM1251804 | not known | not known | 10 | MV4-11 | male |
GSM1251803 | metastasis | poor | 55 | 1103 | male |
GSM1251802 | metastasis | not known | 60 | 1792 | male |
GSM125180 | not known | poor | 61 | RPMI8226 | male |
GSM1251800 | not known | not known | 65 | OCI-AML2 | male |
GSM1251799 | not known | poor | 50 | LNCAP | male |
GSM1251798 | primary | poor | 59 | 629 | male |
GSM1251797 | not known | poor | 36 | L-363 | female |
GSM1251796 | primary | poor | 54 | 393 | male |
GSM1251795 | primary | poor | 63 | 3011 | male |
GSM1251794 | metastasis | good | 46 | DiFi | female |
GSM1251793 | primary | poor | 34 | 529 | female |
GSM1251792 | metastasis | poor | 59 | 983 | male |
GSM125179 | not known | undifferentiated | 57 | JHH-6 | female |
GSM1251790 | not known | not known | 51 | JHH-4 | male |
GSM1251789 | not known | not known | 57 | JHH-2 | male |
GSM1251788 | not known | poor | 38 | OCUM-1 | female |
GSM1251787 | metastasis | poor | 35 | NUGC-4 | female |
GSM1251786 | not known | poor | 62 | MKN45 | female |
GSM1251785 | not known | moderate | 63 | IM95 | male |
GSM1251784 | not known | poor | 66 | Fu97 | female |
GSM1251783 | not known | not known | 54 | SNU-878 | female |
GSM1251782 | not known | not known | 49 | SNU-761 | male |
GSM125178 | not known | not known | 52 | SNU-739 | male |
GSM1251780 | not known | not known | 43 | SNU-475 | male |
GSM1251779 | not known | not known | 52 | SNU-449 | male |
GSM1251778 | not known | not known | 40 | SNU-423 | male |
GSM1251777 | not known | undifferentiated | 68 | HLE | male |
GSM1251776 | not known | not known | 4 | CCRF-CEM-VCR | female |
GSM1251775 | not known | not known | Not available | SNU-899 | Not available |
GSM1251774 | not known | not known | Not available | SNU-1076 | Not available |
GSM1251773 | not known | poor | 62 | 498 | male |
GSM1251772 | not known | poor | 4 | CCRF-CEM | female |
GSM125177 | not known | not known | 72 | MKN1 | male |
GSM1251770 | not known | good | 39 | MKN7 | male |